Green Solvents For Solid Phase Peptide Synthesis

Tea Bags for Fmoc Solid-Phase Peptide Synthesis: An Example of Circular Economy

Assessing the correlation of microscopy‐based and volumetry‐based measurements for resin swelling in a range of potentia

Organic Solvent

Side-chain thioamides as fluorescence quenching probes.

Design of Peptides to Interfere with the RANK-TRAF6 Pathway: an Integrated Approach

Ziconotide ( ω‐conotoxin MVIIA )—Efficient solid‐phase synthesis of a linear precursor peptide and its strategic native

Design, Synthesis, and Evaluation of Linker-Optimised PSMA-Targeting Radioligands

Water-Based Solid-Phase Peptide Synthesis without Hydroxy Side Chain Protection

Scalable and sustainable DMF-free solid-phase synthesis of liraglutideby 1-tert-butyl-3-ethylcarbodiimide-mediated coupl

The Antimicrobial Peptide Capitellacin: Chemical Synthesis of Analogues to Probe the Role of Disulphide Bridges and Thei

Immune system engagers with tuneable properties

Boron-peptide conjugates with angiopep-2 for boron neutron capture therapy

Dipropylamine for 9-Fluorenylmethyloxycarbonyl (Fmoc) Deprotection with Reduced Aspartimide Formation in Solid-Phase Pep

Solid‐Phase Synthesis of Peptidols via Reductive Cleavage Through a Benzotriazole Linker

Total Synthesis and Antimicrobial Evaluation of Pagoamide A

Solvent–Less Environmentally Benign Amino Ester, Amide, and Peptide Synthesis Enabled by Resonant Acoustic Mixing

Chemoselective Solution-

Challenges and Perspectives in Chemical Synthesis of Highly Hydrophobic Peptides

A novel thiol-labile cysteine protecting group for peptide synthesis based on a pyridazinedione (PD) scaffold

Brønsted Acid–Lewis Acid (BA–LA) Induced Final Deprotection/Peptide Resin Cleavage in Fmoc/<i>t-</i>Bu Solid-Phase Pepti

Synthesis of a burkholdine analogue containing β-hydroxytyrosine

Supplementary material from &quot;Synthesis and radiolabelling of PSMA-targeted derivatives containing GYK/MVK cleavable

Enzymatic and chemical synthesis of new anticoagulant peptides

Fast Solution-Phase and Liquid-Phase Peptide Syntheses (SolPSS and LPPS) Mediated by Biomimetic Cyclic Propylphosphonic

Peptides conjugated to 2-alkoxy-8-oxo-adenine as potential synthetic vaccines triggering TLR7

Circular Aqueous Fmoc/t‐Bu Solid‐Phase Peptide Synthesis

Using ¹⁹F NMR and two‐level factorial design to explore thiol‐fluoride substitution in hexafluorobenzene and

Discovery of Dolastatinol: A Synthetic Analog of Dolastatin 10 and Low Nanomolar Inhibitor of Tubulin Polymerization.

Recent Advances in Ynamide Coupling Reagent

Marine Cyclic Peptides: Antimicrobial Activity and Synthetic Strategies

Antioxidant and anti-aging potential of a peptide formulation (Gal2–Pep) conjugated with gallic acid†

Small animal PET imaging with the 68Ga-labeled pH (low) insertion peptide-like peptide YJL-4 in a triple-negative breast

Replacement of Less-Preferred Dipolar Aprotic and

DSPE-PEG Modification of α-Conotoxin TxID

Acid‐Resistant BODIPY Amino Acids for Peptide‐Based Fluorescence Imaging of GPR54 Receptors in Pancreatic Islets

Synthesis of Peptides by Reactive Extrusion. Application to the Continuous and Solventless Preparation of Aspartame.

Chemical Wastes in the Peptide Synthesis Process and Ways to Reduce Them

Survival motor neuron (SMN) protein

Modification of transmembrane peptides to probe SNARE-induced membrane fusion and cross-presentation of membrane-buried

Targeted Amino Acid Substitutions in a Trichoderma Peptaibol Confer Activity against Fungal Plant Pathogens and Protect

- **DOI:** 10.1002/anie.201711143 - **Authors:** Yu, Jin‐Sheng; Noda, Hidetoshi; Shibasaki, Masakatsu - **Year:** 2018 -

Fluorine-induced polarity increases inhibitory activity of BPTI towards chymotrypsin

Identifying the Cellular Target of Cordyheptapeptide A and Synthetic Derivatives.

A Targeted Drug Delivery Strategy for Trypanosomiasis Towards a Diastereoselective Boronate Ester Mediated Intramolecula

<i>N</i>‐ to <i>C</i>‐Peptide Synthesis, Arguably the Future for Sustainable Production

Photo-initiated ring-opening polymerization of N- carboxyanhydrides and its potential application in photolithography

Upscaled Synthesis of α‐ and β‐Peptides in a Continuous‐Flow Reactor Using Propylene Carbonate as an Eco‐Friendly Solven

Chemische Synthese eines SemiSWEET-Transporters

Modulating the Fibrillization of Parathyroid-Hormone (PTH) Peptides: Azo-Switches as Reversible and Catalytic Entities

Toward sustainable solid-phase peptide synthesis strategy – <i>in situ</i> Fmoc removal

Selective Native

A Highly Efficient Synthesis of Polyubiquitin Chains

Constructing nanostructures with atomic precision: The synthesis of spiroligomer-based macrocycles

Morpholine, a strong contender for Fmoc removal in solid‐phase peptide synthesis

Oxetane-based peptidomimetics

Biocompatible strategies for peptide macrocyclisation

Supplementary material from &quot;Phenothiazine-linked Glutamic Acid Dendrons: An Easy Access and a New Class of SARS-Co

New green base for Fmoc removal in solid-phase peptide synthesis: 1,5-diazabicyclo[4.3.0]non-5-ene (DBN), a promising su

Total Synthesis of Scytonemide A Employing Weinreb AM Solid-Phase Resin.

Anti-Cancer Peptides: Status and Future Prospects

Synthèse, analyses structurales et assemblage de foldamères oligoamide hydrosolubles à base de quinolines

Synthesis of Glucosyl Amino Acid Derivatives for Obtaining N‐Glucopeptides via SPPS: Optimization of the Synthetic Route

Study of Novel Peptides for Antimicrobial Protection in Solution and on Cotton Fabric

Analogs of a Natural Peptaibol Exert Anticancer Activity in Both Cisplatin- and Doxorubicin-Resistant Cells and in Multi

The tea-bag protocol for comparison of Fmoc removal reagents in solid-phase peptide synthesis

Improving the Sustainability of Peptide and Polymer Chemistry

Triethyl phosphate (TEP) as a green solvent for solid-phase peptide synthesis (SPPS)

Supplementary material from &quot;Synthesis and radiolabelling of PSMA-targeted derivatives containing GYK/MVK cleavable

(E)-Ethyl-2-cyano-2-(((2,4,6-trichlorobenzoyl)oxy)imino)acetate: A Modified Yamaguchi Reagent for

Synthesis and characterisation of fluorinated molecules that have diverse applications in biology

Propylphosphonic Anhydride (T3P®) as Coupling Reagent for Solid‐Phase Peptide Synthesis

Design and synthesis of novel prodrugs to modulate GABA receptors in cancer

Experimental and Theoretical Screening for Green Solvents Improving Sulfamethizole Solubility

Synthesis of Cyclopeptides

Supplementary material from &quot;Macrocylases as synthetic tools for ligand synthesis: enzymatic synthesis of cyclic pe

Two-helix supramolecular proteomimetic binders assembled via PNA-assisted disulfide crosslinking

N- to C-Peptide Synthesis, Arguably the Future for Sustainable Production

Synthesis of U-theraphotoxin-Pv1a_1, an Aedes aegypti larvicidal disulfide bridged peptide from the Colombian tarantula

Reactor Effluent Compression in a Novel Cyclopentyl Methyl Ether Production Process: A Case Study

Synthesis and Purification of Homogeneous Lipid-Based

Se-Glargine II. Native Function of a Basal Insulin Analog Stabilized by an Internal Diselenide Bridge

A novel approach to amino acid synthesis: acid-assisted reactions with dimethyl carbonate for efficient <i>O</i>-methyla

Amino Acid Composition drives Peptide Aggregation: Predicting Aggregation for Improved Synthesis

Removal of acid-labile protecting or anchoring groups in the presence of polyfluorinated alcohol: Application to solid-p

Sustainable Peptide Synthesis by Photoredox-Catalyzed Picoc-SPPS.

Sulfur And Selenium In Peptides And Proteins: Part I – Chemoselective Methods For Disulfide Bond Formation, Part Ii – Fu

Greening the Solid-Phase Peptide Synthesis Process. 2-MeTHF for the Incorporation of the First Amino Acid and Precipitat

Design, synthesis, and biological evaluation of a multifunctional neuropeptide-Y conjugate for selective nuclear deliver

Linear Peptide Analogues from Jatropha’s Orbitides Promote Migration of Human Neonatal Foreskin Fibroblasts in vitro and

Synthesis and Applications of Porphyrin-Biomacromolecule Conjugates

Amino Acid–Viologen

Synthesis and cellular penetration properties of new phosphonium based cationic amphiphilic peptides† †Electronic supple

Improved Fmoc‐solid‐phase peptide synthesis of an extracellular loop of CFTR for antibody selection by the phage display

<i>N</i>‐Butylpyrrolidinone for Solid‐Phase Peptide Synthesis is Environmentally Friendlier and Synthetically Better tha

Synthetic studies with the brevicidine and laterocidine lipopeptide antibiotics including analogues with enhanced proper

Bike peptides: a ride through the membrane

Triethyl phosphate (TEP) as a green solvent for solid-phase peptide synthesis (SPPS)

OPCML-GPI mimetics as potential biological therapeutics for ovarian cancer

Macromolecular toolbox to elucidate CLE-RLK binding, signaling and downstream effects

Development of lisinopril radioconjugates for nuclear imaging of the angiotensin converting enzyme

Novel amino‐Li resin for water‐based solid‐phase peptide synthesis

Automated solid‐phase synthesis of metabolically stabilized triazolo‐peptidomimetics

Macrocyclisation of small peptides enabled by oxetane incorporation†

The 9-Fluorenylmethoxycarbonyl (Fmoc) Group in Chemical Peptide Synthesis – Its Past, Present, and Future

Small

Scope and Limitations of γ-Valerolactone (GVL) as a Green Solvent to be Used with Base for Fmoc Removal in Solid Phase P

- **DOI:** 10.26262/heal.auth.ir.347860 - **Authors:** Γιαννόπουλος-Δημητρίου, Αλέξανδρος του Δημητρίου - **Year:** 2023

Multimaterial 3D Laser Printing of Cell-Adhesive and Cell-Repellent Hydrogels [data]

Advancing Sustainable Synthesis of Cyclic Peptides by Integrating Aqueous Fmoc/

Refractive Index: The Ultimate Tool for Real-Time Monitoring of Solid-Phase Peptide Synthesis. Greening the Process

Cyclopentyl Methyl Ether (CPME): A Versatile Eco‐Friendly Solvent for Applications in Biotechnology and Biorefineries

Solid‐Phase Synthesis of the Aged‐Nonapeptide‐Nerve‐Agent Adduct of Butyrylcholinesterase as Reference Materials for Ana

Total Synthesis and Bioactivity Mapping of Geodiamolide H

A Diphenylalanine Based Pentapeptide with Fibrillating Self-Assembling Properties

Design of PSMA ligands with modifications at the inhibitor part: an approach to reduce the salivary gland uptake of radi

Preparation, Radiolabeling with 68Ga/177Lu and Preclinical Evaluation of Novel Angiotensin Peptide Analog: A New Class o

SYNTHESIS OF EDEINE DERIVATIVES AS AN APPROACH TO TACKLE THE ANTIBIOTIC CRISIS

Head-to-tail cyclization of side chain-protected linear peptides to recapitulate genetically-encoded cyclized peptides.

Updating the Rulebook: Sustainable Methods for the Construction and Functionalization of Small Molecules Utilizing Micel

Increasing the Functional Group Diversity in Helical β-Peptoids: Achievement of Solvent- and pH-Dependent Folding

Synthesis and Biological Studies of New Temporin A Analogs Containing Unnatural Amino Acids in Position 7

Design, synthesis and structure-activity relationship study of wollamide B; a new potential anti TB agent

Characterization of Synthetic Peptides for Use as an Artificial Oxygen Transporting Material

Studies of Coupling Kinetics and Correlation of Reaction Conversions to Color Tests for Solid-Phase Peptide Synthesis of

การสังเคราะห์ bismacrocyclic SFTI-1 inhibitor และอนุพันธ์

Unveiling the quaternary carbodiimide symphony: harmonizing green chemistry in peptide synthesis

Investigation of Parameters that Affect Resin Swelling in Green Solvents

New green base for Fmoc removal in solid-phase peptide synthesis: 1,5-diazabicyclo[4.3.0]non-5-ene (DBN), a promising su

An explorative study towards the chemical synthesis of the immunoglobulin G1 Fc CH3 domain

Synthesis And Evaluation Of Peptides and Self-Assembled Peptides For Therapeutical Applications

Fluorescent Antibiotics: Bridging Diagnostic and Therapy in the Fight against Bacterial Infections

Integration of DOTA as a bridging unit during solid-phase peptide synthesis

New Temporin A Analogues Modified in Positions 1 and 10—Synthesis and Biological Studies

Design of Peptides for Inhibiting Amyloidogenesis by Blocking Hydrophobic Interactions

Design of an Ultra-Stable Insulin/Glucagon Fusion Protein

Triethyl phosphate (TEP) – dimethylsulfoxide (DMSO), as a green solvent mixture for solid-phase peptide synthesis (SPPS)

Green Solid-Phase Peptide Synthesis (GSPPS) 3. Green Solvents for Fmoc Removal in Peptide Chemistry

Synthesis, Antitumor and Antibacterial Studies of New Shortened Analogues of (KLAKLAK)2-NH2 and Their Conjugates Contain

An optimized protocol for the synthesis of peptides containing trans-cyclooctene and bicyclononyne dienophiles as useful

A novel series of dipeptide derivatives containing indole-3-carboxylic acid conjugates as potential antimicrobial agents

Exploring the Chemical Properties and Medicinal Applications of Tetramethylthiocycloheptyne Sulfoximine Used in Strain-P

Unveiling the quaternary carbodiimide symphony: harmonizing green chemistry in peptide synthesis

Optimized SPPS Process for Octreotide: Using Green Solvent GVL to Reduce Hazardous DMF and Ether Consumption

A Novel Amphibian Antimicrobial Peptide, Phylloseptin-PV1, Exhibits Effective Anti-staphylococcal Activity Without Induc

Development of an in vitro aggregation assay for long synthetic polypeptide, amyloidogenic gelsolin fragment AGelD187N 1

Triptycene: A Nucleic Acid Three-Way Junction Binder Scaffold

Bioinformatics Natural Product Inspired Cyclic Peptides with Diverse Bioactivities

Combining Real-Time Monitoring Using Raman Spectroscopy, Rotating-Bed Reactors, and Green Solvents to Improve Sustainabi

Propylphosphonic anhydride (T3P) as green coupling reagent for solid-phase peptide synthesis

Fundamental Aspects of SPPS and Green Chemical Peptide Synthesis

Any Way You Want It: Pushing the Limits of Chemical Protein Synthesis

Triethyl phosphate (TEP) – dimethylsulfoxide (DMSO), as a green solvent mixture for solid-phase peptide synthesis (SPPS)

Lipodepsipeptide Antibiotics: Total Synthesis and Mechanism of Action Studies Using 19F-NMR

Aspartimide Formation and Its Prevention in Fmoc Chemistry Solid Phase Peptide Synthesis

Imidazole-rich copper peptides as catalysts in xenobiotic degradation

Supplementary material from &quot;Phenothiazine-linked Glutamic Acid Dendrons: An Easy Access and a New Class of SARS-Co

Amino Acid Composition drives Peptide Aggregation: Predicting Aggregation for Improved Synthesis

1,3,5-Triazine as Branching Connector for the Construction of Novel Antimicrobial Peptide Dendrimers: Synthesis and Biol

RGD-functionalized electrospun scaffold for ACL tissue engineering

Small Fluorogenic Amino Acids for Peptide‐Guided Background‐Free Imaging

Synthesis, Antimalarial Activity and Molecular Dynamics Studies of Pipecolisporin: A Novel Cyclic Hexapeptide with Poten

An Efficient, Site‐Selective and Spontaneous Peptide Macrocyclisation During in vitro Translation

- **DOI:** 10.1002/ange.201711143 - **Authors:** Yu, Jin‐Sheng; Noda, Hidetoshi; Shibasaki, Masakatsu - **Year:** 2018 -

<i>N</i>,<i>N</i>‐Dimethyl Formamide European Restriction Demands Solvent Substitution in Research and Development

Supplementary material from &quot;Macrocylases as synthetic tools for ligand synthesis: enzymatic synthesis of cyclic pe

Peptidic Antifreeze Materials: Prospects and Challenges

Greener Cleavage of Protected Peptide Fragments from Sieber Amide Resin

Triethyl phosphate (TEP) – dimethylsulfoxide (DMSO), as a green solvent mixture for solid-phase peptide synthesis (SPPS)

Boc Solid-Phase Synthesis of Conjugable Cyclic Depsipeptide Cotransin for Use as a Biological Probe

Mimicry of Dopamine 1 Receptor Signaling with Cell-Penetrating Peptides

A traceless catch‐and‐release method for rapid peptide purification

Investigation of commercially available resins for the automated flow synthesis of difficult or long peptide sequences

A Peptide-Based Nanocarrier for an Enhanced Delivery and Targeting of Flurbiprofen into the Brain for the Treatment of A

An Atom-Economic Inverse Solid-Phase Peptide Synthesis Using Bn or BcM Esters of Amino Acids

Stereorandomized Oncocins with Preserved Ribosome Binding and Antibacterial Activity.

Development of a novel, automated, robotic system for rapid, high-throughput, parallel, solid-phase peptide synthesis

Scope and Limitations of the Use of Methanesulfonic Acid (MSA) as a Green Acid for Global Deprotection in Solid‐Phase Pe

Facile Protocol for the Synthesis of Self-assembling Polyamine-based Peptide Amphiphiles (PPAs) and Related Biomaterials

Linear Peptide Analogues from Jatropha’s Orbitides Promote Migration of Human Neonatal Foreskin Fibroblasts in vitro and

Synthesis of Cyclic Peptides in SPPS with Npb-OH Photolabile Protecting Group

Process Mass Intensity

Application of a new green protocol in solid-phase peptide synthesis: identification of a new green solvent mixture comp

Safety‐catch linkers for Fmoc solid‐phase synthesis of peptide thioesters and hydrazides by amide‐to‐imide activation

Application of a new green protocol in solid-phase peptide synthesis: identification of a new green solvent mixture comp

Bioinformatics Natural Product Inspired Cyclic Peptides with Diverse Bioactivities

Correction: Synthetic ramoplanin analogues are accessible by effective incorporation of arylglycines in solid-phase pept

Progress Toward Controlled Disulfide Formation To Access Neuroactive Conotoxins

Peptide-EBXs: Enabling Peptide Functionalization and Macrocyclization

Organocatalyst Enabled Light Accelerated Amide and Peptide Synthesis

Synthesis of PNGase-resistant <i>N</i>-glycopeptide containing an α-anomeric glycosidic linkage

A Chemical Biology Approach to Understanding Molecular Recognition of Lipid II by Nisin(1–12): Synthesis and NMR Ensembl

A Shelf Stable Fmoc Hydrazine Resin for the Synthesis of Peptide Hydrazides

Glycoprotein D peptide-based diagnostic approach for the detection of avian infectious laryngotracheitis antibodies

Benzoisothiazolone (BIT): A Fast, Efficient, and Recyclable Redox Reagent for Solid Phase Peptide Synthesis

Green Solid-Phase Peptide Synthesis 2. 2-Methyltetrahydrofuran and Ethyl Acetate for Solid-Phase Peptide Synthesis under

Reflections on a Copenhagen–Minneapolis Axis in Bioorganic Chemistry

Preparação de ésteres de peptídeos através de solvólise e aminólise de peptidil-resinas de kaiser assistidas por Ca<sup>

Automated Glycan Assembly in a Variable-Bed Flow Reactor

Chemical Synthesis of Modularly Modified Analogs of E2/NS1 Peptides on a Novel Chemically and Mechanically Stable Terpol

Rhodiasolv PolarClean – a greener alternative in solid-phase peptide synthesis

Histidine-based copper tetrapeptides as enantioselective catalysts for aldol reactions†

Application of a new green protocol in solid-phase peptide synthesis: identification of a new green solvent mixture comp

<i>N</i>‐Butylpyrrolidinone is an equally good solvent as <i>N</i>,<i>N</i>‐dimethylformamide for microwave assisted sol

Optimization of linker system of potential melanoma skin cancer probe

Solid‐Phase Peptide Macrocyclization and Multifunctionalization via Dipyrrin Construction

Design, Synthesis, and Biological Evaluation of New Analogs of Aurein 1.2 Containing Non-Proteinogenic Amino Acids

2-Methyltetrahydrofuran and cyclopentyl methyl ether for green solid-phase peptide synthesis

Design of PSMA ligands with modifications at the inhibitor part: an approach to reduce the salivary gland uptake of radi

Synthesis of Fmoc-Triazine Amino Acids and Its Application in the Synthesis of Short Antibacterial Peptidomimetics

4-Thioribose Analogues of Adenosine Diphosphate Ribose (ADPr) Peptides.

Synthesis, Characterization and Biomedical Potential of Peptide-Gold Nanoparticle Hydrogels

Synthesis of the Antimicrobial Peptide Murepavadin Using Novel Coupling Agents

A Rapid and Efficient Building Block Approach for Click Cyclization of Peptoids

Synthesis of Peptide N-Acylpyrroles via Anodically Generated N,O-Acetals

Self-assembled proteomimetic (SAP) with antibody-like binding from short PNA–peptide conjugates

Studies of highly N-methylated cyclodepsipeptides, the aureobasidins

Towards the production of tikitericin: A novel peptide from Thermogemmatispora strain T81

Synthesis of the transmembrane domain of the spike protein from SARS‐CoV‐2 using solid phase peptide synthesis and deter

Cyanosulfurylides (CSY): Carboxylic Acid Protecting Groups That Prevent Aspartimide Formation During Peptide Synthesis

Design, synthesis, and biological evaluation of a multifunctional neuropeptide-Y conjugate for selective nuclear deliver

Synthesis of Trifluoromethyl Ketone Containing Amino Acid Building Blocks for the Preparation of Peptide-Based Histone D

Naturally Inspired Peptide Leads: Alanine Scanning Reveals an Actin‐Targeting Thiazole Analogue of Bisebromoamide

Optimized SPPSProcess for Octreotide: Using GreenSolvent GVL to Reduce Hazardous DMF and Ether Consumption

Beyond Efficacy: Ensuring Safety in Peptide Therapeutics through Immunogenicity Assessment

Imidazole-rich copper peptides as catalysts in xenobiotic degradation

Synthese und Anwendung von exo-Methylen-γ-butyrolactonen als potenzielle zytotoxische, carriergebundene Agenzien.

Venomous gland transcriptome and venom proteomic analysis of the scorpion Androctonus amoreuxi reveal new peptides with

Small Fluorogenic Amino Acids for Peptide‐Guided Background‐Free Imaging

Rational design of highly stabilized and selective adrenomedullin analogs

Green solid-phase peptide synthesis 4. γ-Valerolactone and N -formylmorpholine as green solvents for solid phase peptide

Molecular Tools for the Study of ADP-Ribosylation: A Unified and Versatile Method to Synthesise Native Mono-ADP-Ribosyla

Inhibition of jack bean urease by amphiphilic peptides

Synthesis of <i>C</i>‐Glycosyl Amino Acid Building Blocks Suitable for the Solid‐Phase Synthesis of Multivalent Glycopep

Deprotection Bases as an Alternative to the Traditional Bases Used in Solid-Phase Peptide Synthesis

Synthesis of a Fluorescently Tagged Bioactive Probe Specific to Neutrophils in a Zebrafish Model

Novel heterocyclic peptides as potential inhibitors of proteases

<i>N</i>-Butylpyrrolidinone as Alternative Solvent for Solid-Phase Peptide Synthesis

Chemical Synthesis of Six‐Atom Thioether Bridged Diaminodiacid for Solid‐Phase Synthesis of Peptide Disulfide Bond Mimic

The Development of Peptide Ligands to Target H69 rRNA

Synthesis and characterization of time-resolved lanthanide (III) luminescent probes for potential detection of melanoma

Rapid building block-economic synthesis of long, multi-O-GalNAcylated MUC5AC tandem repeat peptides

TIDES unveiled: pioneering green peptides synthesis and oligonucleotides innovations in science

γ-Valerolactone (GVL): An eco-friendly anchoring solvent for solid-phase peptide synthesis

Pyrrole-Mediated Peptide Cyclization Identified through Genetically Reprogrammed Peptide Synthesis

Synthesis, Physicochemical Characterization, In Vitro 2D/3D Human Cell Culture, and In Vitro Aerosol Dispersion Performa

Improved synthesis on solid phase of dithiocarbamic cRGD ‐derivative and ^99mTc ‐radiolabelling

Perfluorophenyl Derivatives as Unsymmetrical Linkers for Solid Phase Conjugation

Progress in Chemical Synthesis of Peptides and Proteins

Design, synthesis, and biological evaluation of a multifunctional neuropeptide-Y conjugate for selective nuclear deliver

Side-Chain Unprotected Fmoc-Arg/His/Tyr-OH Couplings and Their Application in Solid-Phase Peptide Synthesis through a Mi

Toward sustainable solid-phase peptide synthesis strategy – <i>in situ</i> Fmoc removal

Natural Plasmodium falciparum Infection Stimulates Human Antibodies to MSP1 Epitopes Identified in Mice Infection Models

Fully automated synthesis of triazolopeptidomimetics

Total synthesis of a peptide diatom sex pheromone bearing an unusual sulfated aspartic acid

Peptides with 6-Aminohexanoic Acid: Synthesis and Evaluation as Plasmin Inhibitors

Small peptide-based GLP-1R ligands: an approach to reduce the kidney uptake of radiolabeled GLP-1R-targeting agents?

Ultrasonic-Assisted Solid-Phase Peptide Synthesis of DOTA-TATE and DOTA-<i>linker</i>-TATE Derivatives as a Simple and L

Structure-function relationships of disulfide-rich peptides

Targeting tyrosine: a catch-and-release approach to protein modification

Fluorine-induced polarity increases inhibitory activity of BPTI towards chymotrypsin†

Structural Design and Synthesis of Novel Cyclic Peptide Inhibitors Targeting Mycobacterium tuberculosis Transcription

Cover Feature: Upscaled Synthesis of α‐ and β‐Peptides in a Continuous‐Flow Reactor Using Propylene Carbonate as an Eco‐

Small animal PET imaging with the 68Ga-labeled pH (low) insertion peptide-like peptide YJL-4 in a triple-negative breast

Structure-Function Studies of Polymyxin B Lipononapeptides

Synthesis, Antiproliferative Effect and In Silico LogP Prediction of BIM-23052 Analogs Containing Tyr Instead of Phe

Discovery of Selective β-Secretase (BACE-1) Inhibitors by the Solid-Phase Synthesis of Small Molecular-sized Peptides

Silica‐Assisted Solid‐Phase Peptide Synthesis (SiPPS)

Aqueous Solid-Phase Peptide Synthesis (ASPPS) using Standard Fmoc/tBu-Protected Amino Acids

The

Anion binding by fluorescent Fmoc-protected amino acids

Total synthesis of a peptide diatom sex pheromone bearing an unusual sulfated aspartic acid

Revisiting NO2 as Protecting Group of Arginine in Solid-Phase Peptide Synthesis

Synthesis of epitope-tagged venom peptide probes targeting NaV1.7

Ynamide Coupling Reagents: Origin and Advances.

A straightforward method to prevent the under-estimated problem of aspartimide formation during chemical ligation-mediat

Small peptide-based GLP-1R ligands: an approach to reduce the kidney uptake of radiolabeled GLP-1R-targeting agents?

The application of anisole in greener solid-phase peptide synthesis protocols – Compatibility with green bases in Fmoc r

Solid-State Nuclear Magnetic Resonance of Protein Characterization at Fast Magic Angle Spinning

Catalytic and Sustainable Amide Bond Formation using a DABCO/Dichlorotriazine System

Environmentally Friendly SPPS II: Scope of Green Fmoc Removal Protocol Using NaOH and Its Application for Synthesis of C

Triethyl phosphate (TEP) as a green solvent for solid-phase peptide synthesis (SPPS)

Acetyl group for proper protection of β-sugar-amino acids used in SPPS

Evaluation of unexpected protecting group removal in solid‐phase peptide synthesis: Quantified using continuous flow met

Microwave-Assisted Green Solid-Phase Peptide Synthesis Using γ-Valerolactone (GVL) as Solvent

Heptadentate chelates for 89Zr-radiolabelling of monoclonal antibodies†

Synthesis, identification, and characterization ofpeptide natural products and non-natural derivatives

Synthesis and Structural Confirmation of PyHOPO and its Applicability in Racemization Reduction in Solid-Phase Peptide S

Amide Bonds Meet Flow Chemistry: A Journey into Methodologies and Sustainable Evolution

Cyrene: A Green Solvent for the Synthesis of Bioactive Molecules and Functional Biomaterials

Discovery of extended product structural space of the fungal dioxygenase AsqJ

New green base for Fmoc removal in solid-phase peptide synthesis: 1,5-diazabicyclo[4.3.0]non-5-ene (DBN), a promising su

Synthesis of peptides by reactive extrusion. Application to the continuous and solventless preparation of aspartame.

Improving Fmoc Solid Phase Synthesis of Human Beta Defensin 3

Supplementary material from &quot;Totally synthetic microperoxidase-11&quot;

Evaluating the In Vitro Activity

Bioactivity improvement via display of the hydrophobic core of HYD1 in a cyclic β‐hairpin‐like scaffold, MTI‐101

An Efficient Thiol‐ene Mediated Protocol for Thiolated Peptide Synthesis and On‐Resin Diversification

I. Synthesis and Bioactivity of Novel Proteasome Inhibiting Syrbactins and II. Peptide Assembly by Ligation of Hydroxyl

Quantum Defects as a Toolbox for the Covalent Functionalization of Carbon Nanotubes with Peptides and Proteins

Butylated Neuropeptide Antagonist Targeting Hypoxia-Induced GRPR Overexpression in Small Cell Lung Cancer

Greening the Solid-Phase Peptide Synthesis of the First Bicyclic Analogue of the Arc Repressor and Its Binding to DNA

Recent Progress on Green Methods and Technologies for Efficient Formation of Amide Bonds

Dimethyl carbonate as a non-innocent benign solvent for the multistep continuous flow synthesis of amino alcohols

Green Transformation of Solid-Phase Peptide Synthesis

Sustainable Approaches in Solid-phase Peptide Synthesis (SPPS)

Rhodiasolv PolarClean – a greener alternative in solid-phase peptide synthesis

Optimization of peptide synthesis time and sustainability using novel eco‐friendly binary solvent systems with induction

Structural and functional properties of the Kunitz-type and C-terminal domains of Amblyomin-X supporting its antitumor a

Re-evaluating the stability of COMU in different solvents.

Rhodiasolv PolarClean – a greener alternative in solid-phase peptide synthesis

Three Decades of Amyloid Beta Synthesis: Challenges and Advances

Sustainable Ultrasound-Assisted Solid-Phase peptide synthesis (SUS-SPPS): Less Waste, more efficiency

Self-Assembly of a Novel Pentapeptide into Hydrogelated Dendritic Architecture: Synthesis, Properties, Molecular Docking

Semi-synthetic strategies for the synthesis of post-translationally modified Hsp90 variants

Toward a Green SPPS: The Use of an Innovative Mesoporous pDVB Support for Environmentally Friendly Solvents

Combining flavin photocatalysis with parallel synthesis: a general platform to optimize peptides with non-proteinogenic

Troubleshooting When Using γ-Valerolactone (GVL) in Green Solid-Phase Peptide Synthesis

Supplementary material from &quot;Synthesis and radiolabelling of PSMA-targeted derivatives containing GYK/MVK cleavable