testauth · 875 papers with claims · 443 for outreach · 423 old · 9 reviews
<2016
Filtered out
Self-Assembly of a Novel Pentapeptide into Hydrogelated Dendritic Architecture: Synthesis, Properties, Molecular Docking
Amide Bonds Meet Flow Chemistry: A Journey into Methodologies and Sustainable Evolution
N-Butylpyrrolidinone for Solid-Phase Peptide Synthesis is Environmentally Friendlier and Synthetically Better than DMF.
Circular Aqueous Fmoc/t-Bu Solid-Phase Peptide Synthesis.
Catalytic and Sustainable Amide Bond Formation using a DABCO/Dichlorotriazine System
Cover Feature: Upscaled Synthesis of α‐ and β‐Peptides in a Continuous‐Flow Reactor Using Propylene Carbonate as an Eco‐
A Highly Efficient Synthesis of Polyubiquitin Chains.
Inhibition properties of free and conjugated leupeptin analogues
Assessing the correlation of microscopy-based and volumetry-based measurements for resin swelling in a range of potentia
Greener Cleavage of Protected Peptide Fragments from Sieber Amide Resin
N-Butylpyrrolidinone is an equally good solvent as N,N-dimethylformamide for microwave assisted solid phase peptide synt
Investigation of Parameters that Affect Resin Swelling in Green Solvents.
Optimization of peptide synthesis time and sustainability using novel eco-friendly binary solvent systems with induction
2-Methyltetrahydrofuran and cyclopentyl methyl ether for green solid-phase peptide synthesis.
Efficient oxidation of N-protected tryptophan and tryptophanyl-dipeptides by in situ generated dimethyldioxirane provide
Rational design of highly stabilized and selective adrenomedullin analogs
Solid-Phase Synthesis of Gly-Ψ[CH(CF<sub>3</sub>)NH]-Peptides
Environmentally Friendly SPPS II: Scope of Green Fmoc Removal Protocol Using NaOH and Its Application for Synthesis of C
Combining Real-Time Monitoring Using Raman Spectroscopy, Rotating-Bed Reactors, and Green Solvents to Improve Sustainabi
Development of a novel, automated, robotic system for rapid, high-throughput, parallel, solid-phase peptide synthesis.
Environmentally Sensible Organocatalytic Fmoc/t-Bu Solid-Phase Peptide Synthesis.
Bulk Mixing in a Milligram-Scale Solid Phase Batch Reactor
Optimized SPPS Process for Octreotide: Using Green Solvent GVL to Reduce Hazardous DMF and Ether Consumption
Green Solid-Phase Peptide Synthesis (GSPPS) 3. Green Solvents for Fmoc Removal in Peptide Chemistry
Green Solid-Phase Peptide Synthesis 2. 2-Methyltetrahydrofuran and Ethyl Acetate for Solid-Phase Peptide Synthesis under
The application of anisole in greener solid-phase peptide synthesis protocols – Compatibility with green bases in Fmoc r
Advancing Sustainable Peptide Synthesis by Solvent Quality Control: Understanding and Mitigating Hydroperoxide in 1-Buty
Green Solvent Mixtures for Solid-Phase Peptide Synthesis: A Dimethylformamide-Free Highly Efficient Synthesis of Pharmac
2D green SPPS: green solvents for on-resin removal of acid sensitive protecting groups and lactamization
Environmentally friendly SPPS I. Application of NaOH in 2-MeTHF/methanol for Fmoc removal
Greener solvents for solid-phase synthesis
Sustainable Peptide Synthesis by Photoredox-Catalyzed Picoc-SPPS.
Steps towards sustainable solid phase peptide synthesis: use and recovery of <i>N</i>-octyl pyrrolidone
From green innovations in oligopeptide to oligonucleotide sustainable synthesis: differences and synergies in TIDES chem
Advances in solid-phase peptide synthesis in aqueous media (ASPPS)
Replacing DMF in solid-phase peptide synthesis: varying the composition of green binary solvent mixtures as a tool to mi
Greening the synthesis of peptide therapeutics: an industrial perspective.
In situ Fmoc removal – a sustainable solid-phase peptide synthesis approach
<i>Re</i> Green SPPS: enabling circular chemistry in environmentally sensible solid-phase peptide synthesis
Triethyl phosphate (TEP) – dimethylsulfoxide (DMSO), as a green solvent mixture for solid-phase peptide synthesis (SPPS)
Harnessing polarity and viscosity to identify green binary solvent mixtures as viable alternatives to DMF in solid-phase
Application of a new green protocol in solid-phase peptide synthesis: identification of a new green solvent mixture comp
Rhodiasolv PolarClean – a greener alternative in solid-phase peptide synthesis
The 9-Fluorenylmethoxycarbonyl (Fmoc) Group in Chemical Peptide Synthesis – Its Past, Present, and Future
Triethyl phosphate (TEP) as a green solvent for solid-phase peptide synthesis (SPPS)
Evaluation of greener solvents for solid-phase peptide synthesis
Development of bioactive peptides of cosmetic interest through environmentally sustainable processes
Green solvents and Safe Reagents in SPPS taking advantage of induction heating and automation: synthesis and HPLC-free p
Rapid building block-economic synthesis of long, multi-<i>O</i>-GalNAcylated MUC5AC tandem repeat peptides
SYNTHESIS OF POTENT ANTAGONISTS FOR THE NATRIURETIC PEPTIDE CLEARANCE RECEPTOR
Deprotection Bases as an Alternative to the Traditional Bases Used in Solid-Phase Peptide Synthesis.
Synthesis of Killer T Cell Epitopes for Peptide-Based Vaccine of SARS-CoV-2
Flow-based Methods in Chemical Peptide and Protein Synthesis
Scalable and sustainable DMF-free solid-phase synthesis of liraglutideby 1-tert-butyl-3-ethylcarbodiimide-mediated coupl
Aqueous solid-phase peptide synthesis (ASPPS): A novel concept of peptide synthesis
Carbonyl Sulfide-Mediated Synthesis of Peptides with Amino Acid Ionic Liquids
Synthesis of Pentapeptide FWKVV (Phe-Trp-Lys-Val-Val) and Its Activity as Antioxidants
Bachem – Insights into Innovative and Sustainable Peptide Chemistry and Technology by the Leading Independent Manufactur
Rapid building block-economic synthesis of long, multi-O-GalNAcylated MUC5AC tandem repeat peptides
General Installation of (4H)-Imidazolone cis-Amide Bioisosteres Along the Peptide Backbone
Preparation and Application of Green Sustainable Solvent Cyrene
Synthesis of Cystine-Stabilised Dicarba Conotoxin EpI: Ring-Closing Metathesis of Sidechain Deprotected, Sulfide-Rich Se
Solid phase synthesis of four analogs of amyloid-β(9-16) peptide: MS and FT-IR characterization
Peptides as Therapeutic Agents: Challenges and Opportunities in the Green Transition Era
Silylated Tag-Assisted Peptide Synthesis: Continuous One-Pot Elongation for the Production of Difficult Peptides under E
A Practical Peptide Synthesis Workflow Using Amino-Li-Resin
Solid-Phase Insertion of N-mercaptoalkylglycine Residues into Peptides
Amino-Li-Resin—A Fiber Polyacrylamide Resin for Solid-Phase Peptide Synthesis
Dipropyleneglycol Dimethylether, New Green Solvent for Solid-Phase Peptide Synthesis: Further Challenges to Improve Sust
Peptide synthesis: ball-milling, in solution, or on solid support, what is the best strategy?
Improving 2-Chlorotrityl Chloride (2-CTC) Resin Activation.
Green Chemistry of Minimal-Protection Solid-Phase Peptide Synthesis
Bypassing Osmotic Shock Dilemma in a Polystyrene Resin Using the Green Solvent Cyclopentyl methyl Ether (CPME): A Morpho
Recent Progress on Green Methods and Technologies for Efficient Formation of Amide Bonds
Design and synthesis of novel prodrugs to modulate GABA receptors in cancer
A Targeted Drug Delivery Strategy for Trypanosomiasis Towards a Diastereoselective Boronate Ester Mediated Intramolecula
Oxetane-based peptidomimetics
Triethyl phosphate (TEP) – dimethylsulfoxide (DMSO), as a green solvent mixture for solid-phase peptide synthesis (SPPS)
Solid phase peptide synthesis: new resin and new protecting group.
Peptidic Antifreeze Materials: Prospects and Challenges
Structured cyclic peptide mimics by chemical ligation
Scope and Limitations of Barbituric and Thiobarbituric Amino Acid Derivatives as Protecting Groups for Solid‐Phase Pepti
Solid-phase fluorescent BODIPY–peptide synthesis via in situ dipyrrin construction
Imidazole-rich copper peptides as catalysts in xenobiotic degradation.
Total Synthesis and Antimicrobial Evaluation of Pagoamide A
Embedding Peptides into Synthetic Polymers: Radical Ring-Opening Copolymerization of Cyclic Peptides.
A Versatile "Synthesis Tag" (SynTag) for the Chemical Synthesis of Aggregating Peptides and Proteins.
Stabilization of 310-Helices in Macrocycles Using Dominant Rotor Methodology.
Diselenide-selenoester ligation for chemical protein synthesis.
Investigating a PROTAC approach to NRF2 activation
Expressed protein ligation : methods and protocols
Inhibiting protein-protein interactions in telomeres as an approach to cancer chemotherapy
Peptide-Assisted Intracellular Drug Delivery for Boron Neutron Capture Therapy
Synthesis and Purification of Position 4 Analogs of the Opioid Peptide JVA-4001
Synthesis and Biological Evaluation of Novel TLR2 Agonist-Conjugated Antigenic Peptides for use in Cancer Therapeutics
Synthesis of Nocistatin C-terminal and it's Amide Derivatives as an Opioid Peptide.
Chloroalkene dipeptide isosteres as peptidomimetics.
Synthesis, biological evaluation and preclinical study of a novel 99mTc-peptide: A targeting probe of amyloid-β plaques
Design of peptide-based inhibitor agent against amyloid-β aggregation: Molecular docking, synthesis and in vitro evaluat
Design and synthesis of novel antimicrobial peptide scaffolds.
A novel method to produce synthetic murine CXCL10 for efficient screening of functional variants.
Cost-effective synthesis of a chromogenic substrate for SARS-CoV-2 Mpro and development of a miniaturized high-throughpu
Film-Spotting chiral miniPEG-γPNA array for BRCA1 gene mutation detection.
Synthesis of a GlcNAcylated arginine building block for the solid phase synthesis of death domain glycopeptide fragments
Design, synthesis and biological evaluation of phosphopeptides as Polo-like kinase 1 Polo-box domain inhibitors.
Specific Rosetta-based protein-peptide prediction protocol allows the design of novel cholinesterase inhibitor peptides.
Recent advances in racemic protein crystallography.
Synthesis and biological evaluation of peptide-derived TSLP inhibitors.
Stabilization of hyaluronan-based materials by peptide conjugation and its use as a cell-seeded scaffold in tissue engin
In-vitro evaluation of cationic Lipopeptides as adjuvant candidate for DNA plasmid vaccine.
Synthesis and semisynthesis of selenopeptides and selenoproteins.
Design and synthesis of plant cyclopeptide Astin C analogues and investigation of their immunosuppressive activity.
Generation of a glycosylated asparagine residue through chemoselective acylation of a glycosylhydrazide.
Non-covalent interaction between CA-TAT and calf thymus DNA: Deciphering the binding mode by in vitro studies.
Peptide-based targeted cancer therapeutics: design, synthesis and biological evaluation.
Cyclic N-locked indolicidin analogues with antimicrobial activity: Effect of ring size and fatty acid acylation
Protocol for efficient solid-phase synthesis of peptides containing 1-hydroxypyridine-2-one (1,2-HOPO).
A highly sensitive and selective fluorescent "on-off-on" peptide-based probe for sequential detection of Hg2+
A novel fluorescent chemosensor for detection of Zn(II) ions based on dansyl-appended dipeptide in two different living
Synthetic peptide vaccines targeting SVA elicit robust protective immune responses in swine.
A novel fluorescence sensor for uranyl ion detection based on a dansyl-modified peptide.
Efficient synthesis of a side-chain extended diaminodiacid for solid-phase synthesis of peptide disulfide bond mimics
Synthetic peptides to produce antivenoms against the Cys-rich toxins of arachnids.
Solid-phase peptide synthesis of analogues of the N-terminus A-ring fragment of the lantibiotic nisin: Replacements for
Sustainable Ultrasound-Assisted Solid-Phase peptide synthesis (SUS-SPPS): Less Waste, more efficiency.
Synthetic Proteins behind the Plasma Barrier: Molecular Spies
A Custom-EngineeredWater-Soluble Peptide-Based MacrocyclicPolynuclear Gd<sup>3+</sup>-Chelated Paramagnetic Multimodal C
A Custom-EngineeredWater-Soluble Peptide-Based MacrocyclicPolynuclear Gd<sup>3+</sup>-Chelated Paramagnetic Multimodal C
Chemical Synthesis of Peptides Containing Site-Specific Advanced Glycation Endproducts.
A Custom-EngineeredWater-Soluble Peptide-Based MacrocyclicPolynuclear Gd<sup>3+</sup>-Chelated Paramagnetic Multimodal C
Removable Backbone Modification Method for the Chemical Synthesis of Membrane Proteins.
A Custom-Engineered Water-Soluble Peptide-Based Macrocyclic Polynuclear Gd3+-Chelated Paramagnetic Multimodal Contrast A
A Custom-EngineeredWater-Soluble Peptide-Based MacrocyclicPolynuclear Gd<sup>3+</sup>-Chelated Paramagnetic Multimodal C
Chemical Protein Synthesis with the α-Ketoacid-Hydroxylamine Ligation.
A perfluoroaromatic abiotic analog of H2 relaxin enabled by rapid flow-based peptide synthesis.
Solid-phase synthesis and fluorine-18 radiolabeling of cycloRGDyK.
A rink-amide soluble support: high purity conotoxins and other peptides accessed with minimal reagents.
On-resin synthesis of cyclic peptides via tandem N-to-S acyl migration and intramolecular thiol additive-free native che
1,4-Benzenedimethanethiol (1,4-BDMT) as a scavenger for greener peptide resin cleavages
Directed self-assembly of peptide-diketopyrrolopyrrole conjugates - a platform for bio-organic thin film preparation.
Convergent chemoenzymatic synthesis and biological evaluation of a heparan sulfate proteoglycan syndecan-1 mimetic.
A silyl ether-protected building block for O-GlcNAcylated peptide synthesis to enable one-pot acidic deprotection.
Ring-opening reactions for the solid-phase synthesis of nisin lipopeptide analogues.
Asymmetric synthesis of Fmoc-threo-HOAsn for the total synthesis of nicrophorusamide A.
Structural Design and Synthesis of Novel Cyclic Peptide Inhibitors Targeting Mycobacterium tuberculosis Transcription.
Unlocking the Potential of the Antimicrobial Peptide Gomesin: From Discovery and Structure-Activity Relationships to The
Chemical Synthesis and Functional Analysis of VarvA Cyclotide
Convergent Synthesis of Thioether Containing Peptides.
Insulin Hot-Spot Analogs Formed with N-Methylated Amino Acid Residues Inhibit Aggregation of Native Hormone.
Microfluidic Generation of Amino-Functionalized Hydrogel Microbeads Capable of On-Bead Bioassay.
Scope and Limitations of γ-Valerolactone (GVL) as a Green Solvent to be Used with Base for Fmoc Removal in Solid Phase P
Tea Bags for Fmoc Solid-Phase Peptide Synthesis: An Example of Circular Economy.
Flow-Based Fmoc-SPPS Preparation and SAR Study of Cathelicidin-PY Reveals Selective Antimicrobial Activity.
The Hydrophobicity and Antifungal Potentiation of Burkholdine Analogues.
Synthesis of Cyclic Peptides in SPPS with Npb-OH Photolabile Protecting Group.
A Diphenylalanine Based Pentapeptide with Fibrillating Self-Assembling Properties
Design, Synthesis, and Evaluation of Linker-Optimised PSMA-Targeting Radioligands
Synthesis, Antimalarial Activity and Molecular Dynamics Studies of Pipecolisporin: A Novel Cyclic Hexapeptide with Poten
A Bicyclic Analog of the Linear Peptide Arodyn Is a Potent and Selective Kappa Opioid Receptor Antagonist
Challenges in the Characterization and Purification of (Peptide)n-Calix[4]Resorcinarene Conjugates Synthesized via Thiol
Enhancing the Oral Bioavailability of Glutathione Using Innovative Analogue Approaches.
Development of a Polyclonal Antibody for the Immunoanalysis of Ochratoxin A (OTA) by Employing a Specially Designed Synt
Development of Clarstatin, a Novel Drug Lead for the Therapy of Autoimmune Uveitis.
Synthesis and Biological Studies of New Temporin A Analogs Containing Unnatural Amino Acids in Position 7.
[LLC1 neoantigen dendritic cell vaccination combined with CpG effectively converts "cold" tumors into "ho
Facile Protocol for the Synthesis of Self-assembling Polyamine-based Peptide Amphiphiles (PPAs) and Related Biomaterials
Dynamics, Intermolecular Interactions, and Organization of Transmembrane β-Peptides
Peptidomimetic techniques and their application in the design and synthesis of Kisspeptin analogues
Self-Organization of β-Peptide Nucleic Acid Helices for Membrane Scaffolding
Rational Design, Synthesis, and Evaluation of Inhibitors for the HIV-1 TAT Interacting Protein Tip60
An investigation into the key structural role of glycosylated lysine residues in the collagenous domain of adiponectin,
Approaches to target WD40 proteins and synthesis and evaluation of chemical tools for on-bead screening
Universal Access to Protease Chemiluminescent Probes through Solid-Phase Synthesis.
CLipPA Lipidation in the Synthesis of a New Generation of Polymyxin Analogues
Design of Peptides to Interfere with the RANK-TRAF6 Pathway: an Integrated Approach
Synthesis of Mannosylated Lipopeptides with Receptor Targeting Properties.
A Custom-EngineeredWater-Soluble Peptide-Based MacrocyclicPolynuclear Gd<sup>3+</sup>-Chelated Paramagnetic Multimodal C
A Custom-EngineeredWater-Soluble Peptide-Based MacrocyclicPolynuclear Gd<sup>3+</sup>-Chelated Paramagnetic Multimodal C
Photo-controlled reversible binding between the protein A-derived Z domain and immunoglobulin G.
Synthesis of Cyclic Peptides as Potential Anti-Malarials.
Supramolecular Dipeptide-Based Near-Infrared Fluorescent Nanotubes for Cellular Mitochondria Targeted Imaging and Early
A Custom-EngineeredWater-Soluble Peptide-Based MacrocyclicPolynuclear Gd<sup>3+</sup>-Chelated Paramagnetic Multimodal C
Using Chemical Synthesis to Probe Structure-Activity Relationships of the Glycoactive Bacteriocin Glycocin F.
Synthesis and Chemical Structure of the Cyclic Heptapeptide Stylissamide H.
An Organometallic Isostere of an Amino Acid.
Design and Development of an Organocatalyst for Light Accelerated Amide and Peptide Synthesis.
Traceless Solid-Phase Organic Synthesis.
Peptidic Scaffolds Enable Rapid and Multivariate Secondary Sphere Evolution for an Abiotic Metallocatalyst.
Enantioselective Synthesis and Application of Small and Environmentally Sensitive Fluorescent Amino Acids for Probing Bi
Development of Methods for Convergent Synthesis of Chloroalkene Dipeptide Isosteres and Its Application.
Mimicking of Arginine by Functionalized N(ω)-Carbamoylated Arginine As a New Broadly Applicable Approach to Labeled Bioa
Metal-Binding Q-Proline Macrocycles.
Process Development of a Macrocyclic Peptide Inhibitor of PD-L1.
Advancing Sustainable Synthesis of Cyclic Peptides by Integrating Aqueous Fmoc/t-Bu Solid-Phase Peptide Synthesis with D
Process Mass Intensity (PMI): A Holistic Analysis of Current Peptide Manufacturing Processes Informs Sustainability in P
Sulfonate Derivative of HOAt (CTSOAt) as a Coupling Reagent for the Construction of C-N, C-O, and C-C Bonds.
One Step Synthesis of Fmoc-Aminoacyl-N-alkylcysteine via the Ugi Four-Component Condensation Reaction.
Synthesis of Tetra-ortho-Methoxylated Azobenzene Photoswitches via Sequential Catalytic C-H Activation and Methoxylation
α-Azido Acids in Solid-Phase Peptide Synthesis: Compatibility with Fmoc Chemistry and an Alternative Approach to the Sol
Synthesis and SAR Analysis of Lipovelutibols B and D and Their Lipid Analogues.
Total Synthesis and Antimicrobial Activity of Tumescenamide C and Its Derivatives.
Synthesis and Fluorescent Properties of β-Pyridyl α-Amino Acids.
Multiple Synthetic Routes to the Mini-Protein Omomyc and Coiled-Coil Domain Truncations.
Greening the Solid-Phase Peptide Synthesis of the First Bicyclic Analogue of the Arc Repressor and Its Binding to DNA.
Synthesis of Fmoc-Protected Amino Alcohols via the Sharpless Asymmetric Aminohydroxylation Reaction Using FmocNHCl as th
New Teixobactin Analogues with a Total Lactam Ring.
Synthesis of the Antifungal and Antiviral Cyclic Lipodepsipeptides Verlamelins A and B.
Optimized Fmoc-Removal Strategy to Suppress the Traceless and Conventional Diketopiperazine Formation in Solid-Phase Pep
Synthetic Peptides in Doping Control: A Powerful Tool for an Analytical Challenge
Bioconjugation of Cyclometalated Gold(III) Lipoic Acid Fragments to Linear and Cyclic Breast Cancer Targeting Peptides.
Development of High-Functionality and -Quality Lipids with RGD Peptide Ligands: Application for PEGylated Liposomes and
Hybrid Cyclic-Linear Cell-Penetrating Peptides Containing Alternative Positively Charged and Hydrophobic Residues as Mol
Synthesis of a Chloroalkene Dipeptide Isostere-Containing Peptidomimetic and Its Biological Application.
Synthesis of O-Sulfated Human Syndecan-1-like Glyco-polypeptides by Incorporating Peptide Ligation and O-Sulfated Glycop
Synthesis and Purification of Homogeneous Lipid-Based Peptide Nanocarriers by Overcoming Phospholipid Ester Hydrolysis.
Effect of Differences in the Primary Structure of the A-Chain on the Aggregation of Insulin Fragments.
One-Step Synthesis of 3-(Fmoc-amino acid)-3,4-diaminobenzoic Acids.
Hydrophilic Azide-Containing Amino Acid to Enhance the Solubility of Peptides for SPAAC Reactions.
Total Synthesis of Seongsanamide B.
NDTP Mediated Direct Rapid Amide and Peptide Synthesis without Epimerization.
Electrophilic Sulfonium-Promoted Peptide and Protein Amidation in Aqueous Media.
Solid-Phase-Based Synthesis of Lactazole-Like Thiopeptides.
Solid-Phase Total Synthesis of Plusbacin A3.
Spiropyran as Building Block in Peptide Synthesis and Modulation of Photochromic Properties.
Expanding the Reach of Sustainable Solid-Phase Peptide Synthesis: One-Pot, Metal-Free Alloc Removal-Peptide Coupling.
Total Synthesis of a Peptide Diatom Sex Pheromone Bearing a Sulfated Aspartic Acid.
Total Synthesis of LL-A0341β1.
Brønsted Acid-Lewis Acid (BA-LA) Induced Final Deprotection/Peptide Resin Cleavage in Fmoc/t-Bu Solid-Phase Peptide Synt
Total Syntheses of Cyclomarin and Metamarin Natural Products.
N-Sulfanylethylaminooxybutyramide (SEAoxy): A Crypto-Thioester Compatible with Fmoc Solid-Phase Peptide Synthesis.
Chemical Synthesis of HMGA1a Proteins with Post-translational Modifications via Ser/Thr Ligation.
Total Synthesis of Teixobactin.
Synthesis of Oligo-(alkyne-triplet)peptide Constructs.
A Modular and Scalable Route to Protected Cyclopropane Amino Acid Building Blocks.
Synthesis of Insulin-desB30 Analogs via an Enzymatically Removable N-Terminal Solubilizing Tag.
Total Synthesis and Stereochemical Assignment of Gymnopeptides A and B.
An Entirely Solid Phase Peptide Synthesis-Based Strategy for Synthesis of Gelatinase Biosynthesis-Activating Pheromone (
Total Synthesis and Structural Establishment/Revision of Antibiotics A54145.
On-Resin Passerini Reaction toward C-Terminal Photocaged Peptides.
Total Synthesis of Theonellapeptolide Id.
Synthetic α- and β-Ser-ADP-ribosylated Peptides Reveal α-Ser-ADPr as the Native Epimer.
Microwave-Assisted Green Solid-Phase Peptide Synthesis Using γ-Valerolactone (GVL) as Solvent
Solid-Phase Synthesis of Oxetane Modified Peptides.
Synthesis of Chiral Spin-Labeled Amino Acids.
4-Methyltrityl-Protected Pyrrole and Imidazole Building Blocks for Solid Phase Synthesis of DNA-Binding Polyamides.
Chemical Synthesis of K48‐Linked Diubiquitin by Incorporation of a Lysine‐Linked Auxiliary Handle
Tc-99m Glu-Cys-Gly-His-Gly-Lys (ECG-HGK), a novel Tc-99m labeled hexapeptide for molecular tumor imaging.
A novel Tc-99m and fluorescence-labeled arginine-arginine-leucine-containing peptide as a multimodal tumor imaging agent
Synthesis and evaluation of Tc-99m and fluorescence-labeled elastin-derived peptide, VAPG for multimodal tumor imaging i
Dual-labeled prostate-specific membrane antigen (PSMA)-targeting agent for preoperative molecular imaging and fluorescen
Synthesis of carbon-14-labelled peptides.
Gluten Exorphin B5 : Synthesis and Characterization of a Food‐Derived Opioid Peptide
Enzymatically Forming Cell Compatible Supramolecular Assemblies of Tryptophan-Rich Short Peptides.
Bike peptides: a ride through the membrane.
An efficient solid-phase synthesis of peptidyl-N-acetylguanidines for use in native chemical ligation.
Quest for the chemical synthesis of proteins.
Chemical synthesis of N-glycosylated insulin-like androgenic gland factor from the freshwater prawn Macrobrachium rosenb
A comparative study of synthetic and semisynthetic approaches for ligating the epidermal growth factor to a bivalent sca
Complete synthesis of the bicyclic ring of a mutacin analog with orthogonally protected lanthionine via solid-phase intr
Adrenomedullin disulfide bond mimetics uncover structural requirements for AM1 receptor activation.
Antimicrobial activity and secondary structure of a novel peptide derived from ovalbumin.
An explorative study towards the chemical synthesis of the immunoglobulin G1 Fc CH3 domain
Re-evaluating the stability of COMU in different solvents.
Morpholine, a strong contender for Fmoc removal in solid‐phase peptide synthesis
Non‐canonical amino acid bioincorporation into antimicrobial peptides and its challenges
Automated solid-phase synthesis of metabolically stabilized triazolo-peptidomimetics.
Improved Fmoc-solid-phase peptide synthesis of an extracellular loop of CFTR for antibody selection by the phage display
Synthesis of Stylissamide B, a Pro-Rich Cyclic Heptapeptide Isolated From the Marine Sponge Stylissa caribica.
Fundamental Aspects of SPPS and Green Chemical Peptide Synthesis
Structural Modification and Antitumor Activity Study of Peptide Codesane: Discovery of Novel Stapled Peptide Antitumor A
Toward a Green SPPS: The Use of an Innovative Mesoporous pDVB Support for Environmentally Friendly Solvents.
Silica-Assisted Solid-Phase Peptide Synthesis (SiPPS).
Untitled
Design, Synthesis, and Anticancer Activity of N‐1 Terminal Segment of α‐(2, 5,7‐Tri‐tert‐butylindol‐3‐yl)alanine‐Incorpo
Solid‐Phase Microwave‐Assisted Ligand‐Free Suzuki‐Miyaura Cross‐Coupling of 5‐Iodouridine
Evaluation of Anti‐Chlamydial Effect of a Synthetic Linear Peptide
Design of Water-Soluble PEGylated Heptapeptide-Based Multifunctional Magnetic Nanovesicles for Cancer Targeted MRI Integ
Peptidomimetic Synthesis: Drug Discovery for Alzheimer's Disease.
Angiotensin(1-7)-Stearic Acid Conjugate: Synthesis and Characterization
Synthesis of Antioxidant Peptide SCAP1 (Leu-Ala-Asn-Ala-Lys)
Linear Peptide Analogues from Jatropha’s Orbitides Promote Migration of Human Neonatal Foreskin Fibroblasts in vitro and
Development of a KRP-based pH-responsive drug delivery system for solid tumors.
Design of a New 99mTc-radiolabeled Cyclo-peptide as Promising Molecular Imaging Agent of CXCR4 Receptor: Molecular Docki
Prediction of Antithrombin Activity and Bioavailability of a Synthetic Peptide Using a Decision Tree Algorithm.
Modification of the N-Terminus of a Calcium Carbonate Precipitating Peptide Affects Calcium Carbonate Mineralization.
A Novel Dual-labeled Peptide for Multimodal Imaging of EGFR with L858R Mutation.
Total Synthesis of a Reversed-Bacicyclin Using a Combination of Solid- and Solution-Phase Methods
Efficient Synthesis of Norbuprenorphines Coupled with Enkephalins and Investigation of Their Permeability.
Synthesis of Tetrapeptides and Screening of their Antioxidant Properties
Synthesis and evaluation of 99mTc-DOTA-ARA-290 as potential SPECT tracer for targeting cardiac ischemic region.
Production Technology and Functionality of Bioactive Peptides.
Design, Synthesis and Biological Evaluation of Ciprofloxacin- Peptide Conjugates as Anticancer Agents.
1976-LB: A Novel PTAP-009 Peptide—Enhancing Glycemic Control and Sustained Appetite Suppression
Peptidomimetic techniques and their application in the design and synthesis of Kisspeptin analogues
Total Synthesis of the Brevicidine and Laterocidine Family of Lipopeptide Antibiotics
Sintesis Tetrapeptida PSSY dengan Metode Fasa Padat
Total Synthesis of LL-A03411-Beta1
Peptidomimetic techniques and their application in the design and synthesis of Kisspeptin analogues
Traceless Click-Assisted Native Chemical Ligation Enabled by Protecting Dibenzocyclooctyne from Acid-Mediated Rearrangem
An N-terminal selective thiazoline peptide macrocyclisation compatible with mRNA display and efficient SPPS
Design, Synthesis and Labeling of Tripeptide Derivatives with 99mTc as Hypoxia Imaging Agents
Sintesis Tetrapeptida Linier FKAP (Phe-Lys-Ala-Pro) sebagai Kandidat Antioksidan dengan Metode Solid Phase Peptide Synth
Chemical Synthesis of Microtubule-Associated Protein Tau 2N4R
Conjugation of proapoptotic peptides with folate and cyanine dyes for enhanced potency and selectivity towards tumor cel
Polypeptidic Taxol-Tropins: Targeting paclitaxel to the tumor microenvironment
A Benziodoxole-Based Hypervalent Iodine(III) Compound Functioning as a Peptide Coupling Reagent
Histidine 19 Residue Is Essential for Cell Internalization of Antifungal Peptide SmAPα1-21 Derived from the α-Core of th
The Antimicrobial Peptide Capitellacin: Chemical Synthesis of Analogues to Probe the Role of Disulphide Bridges and Thei
Solid Phase Synthesis and TAR RNA-Binding Activity of Nucleopeptides Containing Nucleobases Linked to the Side Chains vi
Natural Cyclic Peptides: Synthetic Strategies and Biomedical Applications
Novel Cyclic Lipopeptide Antibiotics: Effects of Acyl Chain Length and Position.
Fluorescent Analogues of Human α-Calcitonin Gene-Related Peptide with Potent Vasodilator Activity.
Identification, Synthesis, Conformation and Activity of an Insulin-like Peptide from a Sea Anemone.
Development of a Novel Covalently Bonded Conjugate of Caprylic Acid Tripeptide (Isoleucine-Leucine-Aspartic Acid) for Wo
Antimicrobial and Antioxidative Activity of Newly Synthesized Peptides Absorbed into Bacterial Cellulose Carrier against
N-Terminally Lipidated Sialorphin Analogs—Synthesis, Molecular Modeling, In Vitro Effect on Enkephalins Degradation by N
Solid-Phase Synthesis Approaches and U-Rich RNA-Binding Activity of Homotrimer Nucleopeptide Containing Adenine Linked t
Drug Administration Before or After Exposure to Low Temperatures—Does It Matter for the Therapeutic Effect?
Solid-Phase Synthesis of Octapeptin Lipopeptides.
Synthesis of NickFects, a New Family of CPPs, by Solid-Phase Peptide Synthesis.
An Isodipeptide Building Block for Microwave-Assisted Solid-Phase Synthesis of Difficult Sequence-Containing Peptides.
Synthesis of O-Acyl Isopeptides: Stepwise and Convergent Solid-Phase Synthesis.
Solid-Phase Peptide Cyclization with Two Disulfide Bridges.
Synthesis of PNA-Peptide Conjugates as Functional SNARE Protein Mimetics.
Fmoc Solid Phase Peptide Synthesis of Oxytocin and Analogues.
Peptide Hydrazides as Thioester Equivalents for the Chemical Synthesis of Proteins.
Three Methods for Peptide Cyclization Via Lactamization.
Native Chemical Ligation via N-Acylurea Thioester Surrogates Obtained by Fmoc Solid-Phase Peptide Synthesis.
Fmoc Solid-Phase Peptide Synthesis.
Total Linear Chemical Synthesis of LC3A and LC3B.
Removable Backbone Modification (RBM) Strategy for the Chemical Synthesis of Hydrophobic Peptides/Proteins.
Novel Amino-Li Resin for Water-Based Solid-Phase Peptide Synthesis.
Synthesis of Caged Aminoluciferin Peptides.
Improved Handling of Peptide Segments Using Side Chain-Based "Helping Hand" Solubilizing Tools.
Synthesis and Application of SUMO-Based Probes for SUMO Protease Profiling.
Synthesis of Polymyxin-Inspired Peptidomimetics.
Microwave-Assisted Synthesis of Antimicrobial Peptides.
Synthesis of Self-Assembling Peptide-Based Hydrogels for Regenerative Medicine Using Solid-Phase Peptide Synthesis.
Synthesis and Application of Activity-Based Probes for Proteases.
Facile Synthetic Access to Glycopeptide Antibiotic Precursor Peptides for the Investigation of Cytochrome P450 Action in
Thirteen decades of peptide synthesis: key developments in solid phase peptide synthesis and amide bond formation utiliz
Asymmetric synthesis of (2S,3S)-3-Me-glutamine and (R)-allo-threonine derivatives proper for solid-phase peptide couplin
Synthesis and evaluation of tumor-homing peptides for targeting prostate cancer.
A tooth-binding antimicrobial peptide to prevent the formation of dental biofilm.
Citropin 1.1 Trifluoroacetate to Chloride Counter-Ion Exchange in HCl-Saturated Organic Solutions: An Alternative Approa
A novel dual-modality imaging agent targeting folate receptor of tumor for molecular imaging and fluorescence-guided sur
Synthesis and Surface Activity of Cationic Amino Acid‐Based Surfactants in Aqueous Solution
Synthesis and Characterization of Bradykinin Derivatives Based on a β-Cyclodextrin Core
Tc-99m and Fluorescence-Labeled Anti-Flt1 Peptide as a Multimodal Tumor Imaging Agent Targeting Vascular Endothelial Gro
Leveraging the Mukaiyama oxidation-reduction condensation reaction for on-resin aryl thio-esterification for bio-conjuga
Synthesis of Asp-based lactam cyclic peptides using an amide-bonded diaminodiacid to prevent aspartimide formation.
Total synthesis, structure elucidation and expanded bioactivity of icosalide A: effect of lipophilicity and ester to ami
Green solvent mixture for ultrasound-assistant solid-phase peptide synthesis: a fast versatility method and its applicat
Modular solid-phase synthesis of electrophilic cysteine-selective ethynyl-phosphonamidate peptides.
Synthesis of Peptide N-Acylpyrroles via Anodically Generated N,O-Acetals
Synthesis and Structural Stability of α-Helical Gold(I)-Metallopeptidesy
Synthesis of Side-Chain Modified Peptides Using Iterative Solid Phase ‘Click’ Methodology
Retrofitting HPLC Hardware for Affordable and Accessible Flow-Based Peptide Synthesis
Tick saliva protein Evasin-3 modulates chemotaxis by disrupting CXCL8 interactions with glycosaminoglycans and CXCR2
Computational-aided design: minimal peptide sequence to block dengue virus transmission into cells.
Synthesis and Conformational Analysis of APP <i>O</i> ‐Glycopeptides Bearing the Tn Antigen
Synthesis and radiolabelling of PSMA-targeted derivatives containing GYK/MVK cleavable linkers.
A Novel Tumor Imaging Agent, Tc-99m and Fluorescence Labeled Gastrin-Releasing Peptide Analogues
Potential Wound Healing of PLGA Nanoparticles Containing a Novel L ‐Carnitine–GHK Peptide Conjugate
Synergistic antitumor activity of METTL3 peptide degrader and immune checkpoint inhibitor in advanced urothelial cancer.
Introducing Unnatural Amino Acids-Containing Tripeptides as Antimicrobial and Anticancer Agents.
Abstract 4106: A novel synthetic long peptide vaccine composition targeting multiple PD-L1 T-cell epitopes exhibits anti
Enantioselective Synthesis of (2S,3S)‐epi‐Oxetin and Its Incorporation into Conformationally Constrained Pyrrolidinyl PN
Efficient Chemical Protein Synthesis using Fmoc‐Masked N‐Terminal Cysteine in Peptide Thioester Segments
Efficient Chemical Protein Synthesis using Fmoc-Masked N-Terminal Cysteine in Peptide Thioester Segments.
Total Synthesis of α- and β-Amanitin.
Programmable Microwaveable Chemistry in the Chemputer
Leveraging the Knorr Pyrazole Synthesis for the Facile Generation of Thioester Surrogates for use in Native Chemical Lig
Multifunctional peptide-based fluorescent chemosensor for detection of Hg2+ , Cu2+ and S2- ions.
Total Synthesis of Mutanobactins A, B from the Human Microbiome: Macrocyclization and Thiazepanone Assembly in a Single
MgI2 -chemoselective cleavage for removal of amino acid protecting groups: A fresh vision for peptide synthesis.
Side-chain thioamides as fluorescence quenching probes.
Rational Optimizations of the Marine-Derived Peptide Sungsanpin as Novel Inhibitors of Cell Invasion.
Pyrrolidinyl peptide nucleic acids bearing hydroxy-modified cyclobutane building blocks: Synthesis and binding propertie
Designing Chimeric Peptides: A Powerful Tool for Enhancing Antibacterial Activity
Solubilizing Trityl-Type Tag To Synthesize Asx/Glx-Containing Peptides.
B7H6-derived peptides trigger TNF-α-dependent immunostimulatory activity of lymphocytic NK92-MI cells.
Effect of Sulfotyrosine and Negatively Charged Amino Acid of Leech-Derived Peptides on Binding and Inhibitory Activity A
Synthesis of Peptides Containing a Combination of Free and 2-trans-Cyclooctene Carbamate Protected Lysine Residues.
An Efficient, Site‐Selective and Spontaneous Peptide Macrocyclisation During in vitro Translation
Resin Swelling in Mixed Solvents Analysed using Hansen Solubility Parameter Space.
An Optimized Protocol for the Synthesis of Peptides Containing trans-Cyclooctene and Bicyclononyne Dienophiles as Useful
Synthesis of BODIPY-Labeled Cholesterylated Glycopeptides by Tandem Click Chemistry for Glycocalyxification of Giant Uni
Synthesis and Evaluation of Non-Hydrolyzable Phospho-Lysine Peptide Mimics.
Synthesis of l- and d-Ubiquitin by One-Pot Ligation and Metal-Free Desulfurization.
Rapid Chemical Synthesis of Serine Protease Inhibitor Kazal-type 13 (SPINK13) Glycoform by a Combined Method with Glycan
A Tripeptide Approach to the Solid-Phase Synthesis of Peptide Thioacids and N-Glycopeptides.
Synthesis of Asparagine Derivatives Harboring a Lewis X Type DC-SIGN Ligand and Evaluation of their Impact on Immunomodu
Biofunctionalization of Nano Channels by Direct In-Pore Solid-Phase Peptide Synthesis.
Chemical Synthesis of Alpha-Synuclein Proteins via Solid-Phase Peptide Synthesis and Native Chemical Ligation.
A novel Tc-99 m and fluorescence labeled peptide as a multimodal imaging agent for targeting angiogenesis in a murine tu
Scope and Limitations of the Use of Methanesulfonic Acid (MSA) as a Green Acid for Global Deprotection in Solid-Phase Pe
Design, Synthesis, Development, and Biological Evaluation of Third-Generation Tubulin Inhibitors for Treatment of Cancer
Synthesis and Biological Evaluation of Reniochalistatins A-E and a Reniochalistatin E Analogue.
Facile Synthesis of Internal and C‐Terminal Peptide <i>α</i>‐Ketoamides with Fmoc‐Solid Phase Peptide Synthesis
A Custom-EngineeredWater-Soluble Peptide-Based MacrocyclicPolynuclear Gd<sup>3+</sup>-Chelated Paramagnetic Multimodal C
Uniform Preparation of (4R)- and (4S)-Fluoro-l-lysines from One Precursor: Retrosynthesis Software Approach and the Rout
Exploring the Chemical Properties and Medicinal Applications of Tetramethylthiocycloheptyne Sulfoximine Used in Strain-P
Constructing Thioether/Vinyl Sulfide-tethered Helical Peptides Via Photo-induced Thiol-ene/yne Hydrothiolation.
Modification of transmembrane peptides to probe SNARE-induced membrane fusion and cross-presentation of membrane-buried
Cyclization and Derivatization of the Potasium Channel Antagonist Tertiapin
Luminescent Bimetallic Ir III /Au I Peptide Bioconjugates as Potential Theranostic Agents
Sustainable Peptide Synthesis Enabled by a Transient Protecting Group.
Solid-Phase Synthesis of Peptide Hydrazides: Moving Toward Green Chemistry.
Green Solid-Phase Peptide Synthesis: Oxyma-Triggered Spectrophotometric Monitoring of Residual Piperidine
Fmoc-Removal with Pyrrolidine Expands the Available Solvent Space in Green Solid-Phase Peptide Synthesis
Chemical synthesis of membrane proteins by the removable backbone modification method.
Studies Directed Towards the Synthesis of Immunologically Relevant Carbohydrates
Isolation and Structural Elucidation of Antimicrobial Molecules from Crinum ornatum (Aiton) Rhizome of Dutsin-Ma
A Glycyrrhetinic Acid-Modified Curcumin Supramolecular Hydrogel for liver tumor targeting therapy
Chemical synthesis of membrane proteins: a model study on the influenza virus B proton channel.
Stereoselective synthesis of Gly-Gly-type (E)-methylalkene and (Z)-chloroalkene dipeptide isosteres and their applicatio
Epoc group: transformable protecting group with gold(iii)-catalyzed fluorene formation.
Hybrid Cyclic-Linear Cell-Penetrating Peptides Containing Alternative Positive and Hydrophobic Residues as Molecular Tra
Design and Evaluation of Cyclic Peptide-Epirubicin Conjugate for Enhanced Anticancer Activity and Reduced Myocardial Tox
pH- and concentration-dependent supramolecular self-assembly of a naturally occurring octapeptide.
Synthesis and Applications of Synthetic Peptides
Corrigendum: Cross-Talk between Staphylococcus aureus and Other Staphylococcal Species via the agr Quorum Sensing System
Greening Fmoc/tBu solid-phase peptide synthesis
Transport Phenomena in Solid Phase Synthesis Supported by Cross-Linked Polymer Beads
Synthesis of a burkholdine analogue containing β-hydroxytyrosine.
Metal-free photocatalytic cross-electrophile coupling enables C1 homologation and alkylation of carboxylic acids with al
Synthesis of secondary and tertiary amides without coupling agents from amines and potassium acyltrifluoroborates (KATs)
annamaria.papini@unifi.it
Scalable and Sustainable DMF-Free Solid-Phase Synthesis of Liraglutide by 1-Tert-Butyl-3-Ethylcarbodiimide-Mediated Coup
qinsmmu@126.com
pDobz/pDobb protected diaminodiacid as a novel building block for peptide disulfide-bond mimic synthesis.
n.i.martin@biology.leidenuniv.nl
Macrocyclic peptides as allosteric inhibitors of nicotinamide <i>N</i> -methyltransferase (NNMT)
v.chudasama@ucl.ac.uk
A novel thiol-labile cysteine protecting group for peptide synthesis based on a pyridazinedione (PD) scaffold.
gsammis@chem.ubc.ca
Rapid and column-free syntheses of acyl fluorides and peptides using ex situ generated thionyl fluoride.
hagimori@mukogawa-u.ac.jp
Synthesis and physicochemical evaluation of fluorinated lipopeptide precursors of ligands for microbubble targeting.
anahhas@kau.edu.sa
Developing and Testing Methylated Nano-Structured Dipeptides that Inhibit Src Kinase Activity In Vitro for Anti-Cancer A
zhaodx798@163.com
Synthesis and Preliminary Study on the DNA-binding Property of Tranexamic Acid Derivatives
albericio@ukzn.ac.za
Solid-Phase Peptide Synthesis Using a Four-Dimensional (Safety-Catch) Protecting Group Scheme.
frank.boeckler@uni-tuebingen.de
Synthesis of Amino Acids Bearing Halodifluoromethyl Moieties and Their Application to p53-Derived Peptides Binding to Md
koorbanally@ukzn.ac.za
Perfluorophenyl Derivatives as Unsymmetrical Linkers for Solid Phase Conjugation.
walter.cabri@unibo.it
Solid Phase Peptide Synthesis using side-chain unprotected arginine and histidine, with Oxyma Pure/TBEC in green solvent
simona.serban@sunresin.com
Towards green, scalable peptide synthesis: leveraging DEG-crosslinked polystyrene resins to overcome hydrophobicity chal
luciano.lattuada@bracco.com
Improved synthesis of DA364, an NIR fluorescence RGD probe targeting α v β 3 integrin
ron.nachman@usda.gov
Solid Phase Synthesis of an Insect Pyrokinin Analog Incorporating an Imidazoline Ring as Isosteric Replacement of a <em>